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代谢疾病Identifying novel adenosine receptor ligands by simultaneous proteochemometric modeling of rat and human bioactivity data.

期刊:Journal of medicinal chemistry发表年份:2012作者:Gerard J P van Westen; Olaf O van den Hoven; Rianne van der Pijl; Thea Mulder-Krieger; Henk de Vries; Jörg K Wegner; Adriaan P Ijzerman; Herman W T van Vlijmen; Andreas Bender

代谢疾病Design, synthesis, structural and functional characterization of novel melanocortin agonists based on the cyclotide kalata B1.

期刊:The Journal of biological chemistry发表年份:2012作者:Rasmus Eliasen; Norelle L Daly; Birgitte S Wulff; Thomas L Andresen; Kilian W Conde-Frieboes; David J Craik

代谢疾病Structure-activity relationships and key structural feature of pyridyloxybenzene-acylsulfonamides as new, potent, and selective peroxisome proliferator-activated receptor (PPAR) γ Agonists.

期刊:Bioorganic & medicinal chemistry发表年份:2012作者:Kentaro Rikimaru; Takeshi Wakabayashi; Hidenori Abe; Taisuke Tawaraishi; Hiroshi Imoto; Jinichi Yonemori; Hideki Hirose; Katsuhito Murase; Takanori Matsuo; Mitsuharu Matsumoto; Chisako Nomura; Hiroko Tsuge; Naoto Arimura; Kazutoshi Kawakami; Junichi

代谢疾病Evaluation of a 125I-labelled benzazepinone derived voltage-gated sodium channel blocker for imaging with SPECT.

期刊:Organic & biomolecular chemistry发表年份:2012作者:Carlos Pérez-Medina; Niral Patel; Mathew Robson; Adam Badar; Mark F Lythgoe; Erik Årstad