其他Difluoromethylene at the γ-Lactam α-Position Improves 11-Deoxy-8-aza-PGE1 Series EP4 Receptor Binding and Activity: 11-Deoxy-10,10-difluoro-8-aza-PGE1 Analog (KMN-159) as a Potent EP4 Agonist.
期刊:Journal of medicinal chemistry发表年份:2019作者:Stephen D Barrett; Melissa C Holt; James B Kramer; Bradlee Germain; Chi S Ho; Fred L Ciske; Andrei Kornilov; Joseph M Colombo; Adam Uzieblo; James P O'Malley; Thomas A Owen; Adam J Stein; Maria I Morano
