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其他Discovery and in vitro and in vivo profiles of N-ethyl-N-[2-[3-(5-fluoro-2-pyridinyl)-1H-pyrazol-1-yl]ethyl]-2-(2H-1,2,3-triazol-2-yl)-benzamide as a novel class of dual orexin receptor antagonist.

期刊:Bioorganic & medicinal chemistry发表年份:2015作者:Ryo Suzuki; Dai Nozawa; Aya Futamura; Rie Nishikawa-Shimono; Masahito Abe; Nobutaka Hattori; Hiroshi Ohta; Yuko Araki; Daiji Kambe; Mari Ohmichi; Seiken Tokura; Takeshi Aoki; Norikazu Ohtake; Hiroshi Kawamoto

其他Slingshot-Cofilin activation mediates mitochondrial and synaptic dysfunction via Aβ ligation to β1-integrin conformers.

期刊:Cell death and differentiation发表年份:2015作者:J A Woo; X Zhao; H Khan; C Penn; X Wang; A Joly-Amado; E Weeber; D Morgan; D E Kang

其他Constructing de novo H2O2 signaling via induced protein proximity.

期刊:ACS chemical biology发表年份:2015作者:Guihua Zeng; Roushu Zhang; Weimin Xuan; Wei Wang; Fu-Sen Liang

其他Design, synthesis, and biological evaluation of novel 2-((2-(4-(substituted)phenylpiperazin-1-yl)ethyl)amino)-5'-N-ethylcarboxamidoadenosines as potent and selective agonists of the A2A adenosine receptor.

期刊:Journal of medicinal chemistry发表年份:2015作者:Delia Preti; Pier Giovanni Baraldi; Giulia Saponaro; Romeo Romagnoli; Mojgan Aghazadeh Tabrizi; Stefania Baraldi; Sandro Cosconati; Agostino Bruno; Ettore Novellino; Fabrizio Vincenzi; Annalisa Ravani; Pier Andrea Borea; Katia Varani