其他Discovery of 6alpha-ethyl-23(S)-methylcholic acid (S-EMCA, INT-777) as a potent and selective agonist for the TGR5 receptor, a novel target for diabesity.
期刊:Journal of medicinal chemistry发表年份:2009作者:Roberto Pellicciari; Antimo Gioiello; Antonio Macchiarulo; Charles Thomas; Emiliano Rosatelli; Benedetto Natalini; Roccaldo Sardella; Mark Pruzanski; Aldo Roda; Elisabetta Pastorini; Kristina Schoonjans; Johan Auwerx