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基因编辑仓鼠Biased agonism and allosteric modulation of G protein-coupled receptor 183 - a 7TM receptor also known as Epstein-Barr virus-induced gene 2.

期刊:British journal of pharmacology发表年份:2017作者:Viktorija Daugvilaite; Christian Medom Madsen; Michael Lückmann; Clara Castello Echeverria; Andreas Walter Sailer; Thomas Michael Frimurer; Mette Marie Rosenkilde; Tau Benned-Jensen

基因编辑仓鼠Dampened activity of ryanodine receptor channels in mutant skeletal muscle lacking TRIC-A.

期刊:The Journal of physiology发表年份:2017作者:Sam El-Ajouz; Elisa Venturi; Katja Witschas; Matthew Beech; Abigail D Wilson; Chris Lindsay; David Eberhardt; Fiona O'Brien; Tsunaki Iida; Miyuki Nishi; Hiroshi Takeshima; Rebecca Sitsapesan

基因编辑仓鼠Discovery and characterization of a novel irreversible EGFR mutants selective and potent kinase inhibitor CHMFL-EGFR-26 with a distinct binding mode.

期刊:Oncotarget发表年份:2017作者:Chen Hu; Aoli Wang; Hong Wu; Ziping Qi; Xixiang Li; Xiao-E Yan; Cheng Chen; Kailin Yu; Fengming Zou; Wenchao Wang; Wei Wang; Jiaxin Wu; Juan Liu; Beilei Wang; Li Wang; Tao Ren; Shanchun Zhang; Cai-Hong Yun; Jing Liu; Qingsong Liu

基因编辑仓鼠Generic membrane-spanning features endow IRE1α with responsiveness to membrane aberrancy.

期刊:Molecular biology of the cell发表年份:2017作者:Nozomu Kono; Niko Amin-Wetzel; David Ron