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代谢疾病High-throughput screening campaign identifies a small molecule agonist of the relaxin family peptide receptor 4.

期刊:Acta pharmacologica Sinica发表年份:2020作者:Guang-Yao Lin; Lin Lin; Xiao-Qing Cai; An-Tao Dai; Yue Zhu; Jie Li; Qing Liu; De-Hua Yang; Ross A D Bathgate; Ming-Wei Wang

代谢疾病Discovery and Evaluation of Enantiopure 9H-pyrimido[4,5-b]indoles as Nanomolar GSK-3β Inhibitors with Improved Metabolic Stability.

期刊:International journal of molecular sciences发表年份:2020作者:Stanislav Andreev; Tatu Pantsar; Ahmed El-Gokha; Francesco Ansideri; Mark Kudolo; Débora Bublitz Anton; Giulia Sita; Jenny Romasco; Christian Geibel; Michael Lämmerhofer; Márcia Ines Goettert; Andrea Tarozzi; Stefan A Laufer; Pierre Koch

代谢疾病Investigation of the Adrenergic and Opioid Binding Affinities, Metabolic Stability, Plasma Protein Binding Properties, and Functional Effects of Selected Indole-Based Kratom Alkaloids.

期刊:Journal of medicinal chemistry发表年份:2020作者:Samuel Obeng; Shyam H Kamble; Morgan E Reeves; Luis F Restrepo; Avi Patel; Mira Behnke; Nelson J-Y Chear; Surash Ramanathan; Abhisheak Sharma; Francisco León; Takato Hiranita; Bonnie A Avery; Lance R McMahon; Christopher R McCurdy

代谢疾病Identification of potent pyrazole based APELIN receptor (APJ) agonists.

期刊:Bioorganic & medicinal chemistry发表年份:2020作者:Sanju Narayanan; Vineetha Vasukuttan; Sudarshan Rajagopal; Rangan Maitra; Scott P Runyon