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代谢疾病Mono-PEGylates of exenatide in branched and dimeric structures can improve in vivo stability and hypoglycemic bioactivity.

期刊:Journal of biotechnology发表年份:2019作者:Ngoc-Thanh Thi Nguyen; Sujin Jung; Seung Hwan Lee; Ok Nam Bae; E K Lee

代谢疾病The Bioorthogonal Isonitrile-Chlorooxime Ligation.

期刊:Journal of the American Chemical Society发表年份:2019作者:Rebecca J B Schäfer; Mattia R Monaco; Mao Li; Alina Tirla; Pablo Rivera-Fuentes; Helma Wennemers

代谢疾病Discovery of potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor SGL5213 for type 2 diabetes treatment.

期刊:Bioorganic & medicinal chemistry发表年份:2019作者:Shoichi Kuroda; Yohei Kobashi; Takahiro Oi; Kenichi Kawabe; Fumiyasu Shiozawa; Lisa Okumura-Kitajima; Mami Sugisaki-Kitano; Fusayo Io; Koji Yamamoto; Hiroyuki Kakinuma

代谢疾病Molecular Basis of Action of a Small-Molecule Positive Allosteric Modulator Agonist at the Type 1 Cholecystokinin Holoreceptor.

期刊:Molecular pharmacology发表年份:2019作者:Aditya J Desai; Ingrid Mechin; Karthigeyan Nagarajan; Celine Valant; Denise Wootten; Polo C H Lam; Andrew Orry; Ruben Abagyan; Anil Nair; Patrick M Sexton; Arthur Christopoulos; Laurence J Miller