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代谢疾病Transcriptome Analysis of Hypothalamic Gene Expression during Daily Torpor in Djungarian Hamsters (Phodopus sungorus).

期刊:Frontiers in neuroscience发表年份:2017作者:Ceyda Cubuk; Julia Kemmling; Andrej Fabrizius; Annika Herwig

代谢疾病Discovery of a Potent, Selective Renal Sodium-Dependent Glucose Cotransporter 2 (SGLT2) Inhibitor (HSK0935) for the Treatment of Type 2 Diabetes.

期刊:Journal of medicinal chemistry发表年份:2017作者:Yao Li; Zongjun Shi; Lei Chen; Suxin Zheng; Sheng Li; Bo Xu; Zhenhong Liu; Jianyu Liu; Chongyang Deng; Fei Ye

代谢疾病Structural development of 1,2,3,4-tetrahydroisoquinoline-type positive allosteric modulators of prostacyclin receptor (IPPAMs) to improve metabolic stability, and investigation of metabolic fate.

期刊:Bioorganic & medicinal chemistry letters发表年份:2017作者:Hiroyuki Miyachi; Toshifumi Suzuki; Riyo Imamura; Tetsuo Nagano; Takayoshi Okabe

代谢疾病Discovery of novel 5-oxa-2,6-diazaspiro[3.4]oct-6-ene derivatives as potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonists for treatment of type 2 diabetes mellitus.

期刊:Bioorganic & medicinal chemistry发表年份:2017作者:Hideki Hirose; Takeshi Yamasaki; Masaki Ogino; Ryo Mizojiri; Yumiko Tamura-Okano; Hiroaki Yashiro; Yo Muraki; Yoshihide Nakano; Jun Sugama; Akito Hata; Shinji Iwasaki; Masanori Watanabe; Tsuyoshi Maekawa; Shizuo Kasai