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代谢疾病Design, synthesis, and biological evaluation of a novel series of peripheral-selective noradrenaline reuptake inhibitors-Part 2.

期刊:Bioorganic & medicinal chemistry发表年份:2016作者:Tomoya Yukawa; Ikuo Fujimori; Taku Kamei; Yoshihisa Nakada; Nobuki Sakauchi; Masami Yamada; Yusuke Ohba; Hiroyuki Ueno; Maiko Takiguchi; Masako Kuno; Izumi Kamo; Hideyuki Nakagawa; Yasushi Fujioka; Tomoko Igari; Yuji Ishichi; Tetsuya Tsukamoto

代谢疾病Human CB1 Receptor Isoforms, present in Hepatocytes and β-cells, are Involved in Regulating Metabolism.

期刊:Scientific reports发表年份:2016作者:Isabel González-Mariscal; Susan M Krzysik-Walker; Máire E Doyle; Qing-Rong Liu; Raffaello Cimbro; Sara Santa-Cruz Calvo; Soumita Ghosh; Łukasz Cieśla; Ruin Moaddel; Olga D Carlson; Rafal P Witek; Jennifer F O'Connell; Josephine M Egan

代谢疾病Conopeptide-Derived κ-Opioid Agonists (Conorphins): Potent, Selective, and Metabolic Stable Dynorphin A Mimetics with Antinociceptive Properties.

期刊:Journal of medicinal chemistry发表年份:2016作者:Andreas Brust; Daniel E Croker; Barbara Colless; Lotten Ragnarsson; Åsa Andersson; Kapil Jain; Sonia Garcia-Caraballo; Joel Castro; Stuart M Brierley; Paul F Alewood; Richard J Lewis

代谢疾病An AlphaScreen Assay for the Discovery of Synthetic Chemical Inhibitors of Glucagon Production.

期刊:Journal of biomolecular screening发表年份:2016作者:Matthew R Evans; Shuguang Wei; Bruce A Posner; Roger H Unger; Michael G Roth