郑州微飒生物科技有限责任公司 咨询热线:0371-88821766
行业动态

行业动态

追踪行业前沿,洞察产业趋势

代谢疾病N-Indolylglycosides bearing modifications at the glucose C6-position as sodium-dependent glucose co-transporter 2 inhibitors.

期刊:Bioorganic & medicinal chemistry发表年份:2016作者:Kuang-Feng Chu; Chun-Hsu Yao; Jen-Shin Song; Chiung-Tong Chen; Teng-Kuang Yeh; Tsung-Chih Hsieh; Chung-Yu Huang; Min-Hsien Wang; Szu-Huei Wu; Wei-En Chang; Yu-Sheng Chao; Jinq-Chyi Lee

代谢疾病Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139.

期刊:Scientific reports发表年份:2016作者:Mohamed A Shehata; Anne C Nøhr; Delphine Lissa; Christoph Bisig; Vignir Isberg; Kirsten B Andersen; Kasper Harpsøe; Fredrik Björkling; Hans Bräuner-Osborne; David E Gloriam

代谢疾病AZD8797 is an allosteric non-competitive modulator of the human CX3CR1 receptor.

期刊:The Biochemical journal发表年份:2016作者:Linda Cederblad; Birgitta Rosengren; Erik Ryberg; Nils-Olov Hermansson

代谢疾病The C-terminus of the B-chain of human insulin-like peptide 5 is critical for cognate RXFP4 receptor activity.

期刊:Amino acids发表年份:2016作者:Nitin A Patil; Ross A D Bathgate; Martina Kocan; Sheng Yu Ang; Julien Tailhades; Frances Separovic; Roger Summers; Johannes Grosse; Richard A Hughes; John D Wade; Mohammed Akhter Hossain