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代谢疾病Further Optimization and Evaluation of Bioavailable, Mixed-Efficacy μ-Opioid Receptor (MOR) Agonists/δ-Opioid Receptor (DOR) Antagonists: Balancing MOR and DOR Affinities.

期刊:Journal of medicinal chemistry发表年份:2015作者:Aubrie A Harland; Larisa Yeomans; Nicholas W Griggs; Jessica P Anand; Irina D Pogozheva; Emily M Jutkiewicz; John R Traynor; Henry I Mosberg

代谢疾病Novel, potent, selective and cellular active ABC type PTP1B inhibitors containing (methanesulfonyl-phenyl-amino)-acetic acid methyl ester phosphotyrosine mimetic.

期刊:Bioorganic & medicinal chemistry发表年份:2015作者:Peihong Liu; Yongli Du; Lianhua Song; Jingkang Shen; Qunyi Li

代谢疾病Optical Control of Insulin Secretion Using an Incretin Switch.

期刊:Angewandte Chemie (International ed. in English)发表年份:2015作者:Johannes Broichhagen; Tom Podewin; Helena Meyer-Berg; Yorrick von Ohlen; Natalie R Johnston; Ben J Jones; Stephen R Bloom; Guy A Rutter; Anja Hoffmann-Röder; David J Hodson; Dirk Trauner

代谢疾病Role of Δ1-pyrroline-5-carboxylate dehydrogenase supports mitochondrial metabolism and host-cell invasion of Trypanosoma cruzi.

期刊:The Journal of biological chemistry发表年份:2015作者:Brian S Mantilla; Lisvane S Paes; Elizabeth M F Pral; Daiana E Martil; Otavio H Thiemann; Patricio Fernández-Silva; Erick L Bastos; Ariel M Silber