郑州微飒生物科技有限责任公司 咨询热线:0371-88821766
行业动态

行业动态

追踪行业前沿,洞察产业趋势

代谢疾病Can silicon make an excellent drug even better? An in vitro and in vivo head-to-head comparison between loperamide and its silicon analogue sila-loperamide.

期刊:ChemMedChem发表年份:2015作者:Marcel Geyer; Eric Wellner; Ulrik Jurva; Sebastian Saloman; Duncan Armstrong; Reinhold Tacke

代谢疾病Elimination of a cholecystokinin receptor agonist 'trigger' in an effort to develop positive allosteric modulators without intrinsic agonist activity.

期刊:Bioorganic & medicinal chemistry letters发表年份:2015作者:Aditya J Desai; Brad R Henke; Laurence J Miller

代谢疾病Combined Optical Coherence and Fluorescence Microscopy to assess dynamics and specificity of pancreatic beta-cell tracers.

期刊:Scientific reports发表年份:2015作者:Corinne Berclaz; Christophe Pache; Arno Bouwens; Daniel Szlag; Antonio Lopez; Lieke Joosten; Selen Ekim; Maarten Brom; Martin Gotthardt; Anne Grapin-Botton; Theo Lasser

代谢疾病Molecular Mechanism of Action of Triazolobenzodiazepinone Agonists of the Type 1 Cholecystokinin Receptor. Possible Cooperativity across the Receptor Homodimeric Complex.

期刊:Journal of medicinal chemistry发表年份:2015作者:Aditya J Desai; Polo C H Lam; Andrew Orry; Ruben Abagyan; Arthur Christopoulos; Patrick M Sexton; Laurence J Miller