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代谢疾病Optimization of ketone-based P2Y(12) receptor antagonists as antithrombotic agents: pharmacodynamics and receptor kinetics considerations.

期刊:Bioorganic & medicinal chemistry letters发表年份:2014作者:Fabrizio Giordanetto; Peter Bach; Fredrik Zetterberg; Thomas Antonsson; Ruth Bylund; Johan Johansson; Mikael Sellén; David Brown; Lotta Hideståhl; Pia Berntsson; Daniel Hovdal; Helen Zachrisson; Jan-Arne Björkman; J J J van Giezen

代谢疾病Signalling profiles of H3 relaxin, H2 relaxin and R3(BΔ23-27)R/I5 acting at the relaxin family peptide receptor 3 (RXFP3).

期刊:British journal of pharmacology发表年份:2014作者:M Kocan; M Sarwar; M A Hossain; J D Wade; R J Summers

代谢疾病In vitro metabolism of cis- and trans-permethrin by rat liver microsomes, and its effect on estrogenic and anti-androgenic activities.

期刊:Environmental toxicology and pharmacology发表年份:2014作者:Satoko Tange; Nariaki Fujimoto; Naoto Uramaru; Kazumi Sugihara; Shigeru Ohta; Shigeyuki Kitamura

代谢疾病Identification of neuropeptide S antagonists: structure-activity relationship studies, X-ray crystallography, and in vivo evaluation.

期刊:ACS chemical neuroscience发表年份:2014作者:Carla Hassler; Yanan Zhang; Brian Gilmour; Tyler Graf; Timothy Fennell; Rodney Snyder; Jeffrey R Deschamps; Rainer K Reinscheid; Celia Garau; Scott P Runyon