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代谢疾病Synthesis and in vivo evaluation of (S)-6-(4-fluorophenoxy)-3-((1-[11C]methylpiperidin-3-yl)methyl)-2-o-tolylquinazolin-4(3H)-one, a potential PET tracer for growth hormone secretagogue receptor (GHSR).

期刊:Bioorganic & medicinal chemistry发表年份:2011作者:Rachel Potter; Andrew G Horti; Hayden T Ravert; Daniel P Holt; Paige Finley; Ursula Scheffel; Robert F Dannals; Richard L Wahl

代谢疾病Melanin-concentrating hormone receptor 1 antagonists: synthesis, structure-activity relationship, docking studies, and biological evaluation of 2,3,4,5-tetrahydro-1H-3-benzazepine derivatives.

期刊:Bioorganic & medicinal chemistry发表年份:2011作者:Shizuo Kasai; Masahiro Kamaura; Makoto Kamata; Kazuyoshi Aso; Hitomi Ogino; Yoshihide Nakano; Kaoru Watanabe; Tomoko Kaisho; Michiko Tawada; Yasutaka Nagisa; Shiro Takekawa; Koki Kato; Nobuhiro Suzuki; Yuji Ishihara

代谢疾病Dual mode of glucagon receptor internalization: role of PKCα, GRKs and β-arrestins.

期刊:Experimental cell research发表年份:2011作者:Lada Krilov; Amy Nguyen; Teruo Miyazaki; Cecilia G Unson; Russell Williams; Norman H Lee; Susan Ceryak; Bernard Bouscarel

代谢疾病Application of the DNA adductome approach to assess the DNA-damaging capability of in vitro micronucleus test-positive compounds.

期刊:Mutation research发表年份:2011作者:Kyoko Kato; Eiji Yamamura; Masanobu Kawanishi; Takashi Yagi; Tomonari Matsuda; Akio Sugiyama; Yoshifumi Uno