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代谢疾病N-(Pyridin-2-yl) arylsulfonamide inhibitors of 11beta-hydroxysteroid dehydrogenase type 1: Discovery of PF-915275.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Michael Siu; Theodore O Johnson; Yong Wang; Sajiv K Nair; Wendy D Taylor; Stephan J Cripps; Jean J Matthews; Martin P Edwards; Thomas A Pauly; Jacques Ermolieff; Arturo Castro; Natilie A Hosea; Amy LaPaglia; Andrea N Fanjul; Jennifer E Vogel

代谢疾病Discovery of a novel azepine series of potent and selective 5-HT2C agonists as potential treatments for urinary incontinence.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Paul E Brennan; Gavin A Whitlock; Danny K H Ho; Kelly Conlon; Gordon McMurray

代谢疾病Discovery of a peroxisome proliferator activated receptor gamma (PPARgamma) modulator with balanced PPARalpha activity for the treatment of type 2 diabetes and dyslipidemia.

期刊:Journal of medicinal chemistry发表年份:2009作者:Weiguo Liu; Kun Liu; Harold B Wood; Margaret E McCann; Thomas W Doebber; Ching H Chang; Taro E Akiyama; Monica Einstein; Joel P Berger; Peter T Meinke

代谢疾病Metabolic labeling of sialic acids in living animals with alkynyl sugars.

期刊:Angewandte Chemie (International ed. in English)发表年份:2009作者:Pamela V Chang; Xing Chen; Chris Smyrniotis; Alexander Xenakis; Tianshun Hu; Carolyn R Bertozzi; Peng Wu