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药效评价Indoline derivatives I: synthesis and factor Xa (FXa) inhibitory activities.

期刊:Chemical & pharmaceutical bulletin发表年份:2006作者:Tetsuji Noguchi; Naoki Tanaka; Toyoki Nishimata; Riki Goto; Miho Hayakawa; Atsuhiro Sugidachi; Taketoshi Ogawa; Fumitoshi Asai; Yumi Matsui; Koichi Fujimoto

药效评价Synthesis and in vitro pharmacological studies of new C(4)-modified salvinorin A analogues.

期刊:Bioorganic & medicinal chemistry letters发表年份:2006作者:David Y W Lee; Minsheng He; Lee-Yuan Liu-Chen; Yulin Wang; Jian-Guo Li; Wei Xu; Zhongze Ma; William A Carlezon; Bruce Cohen

药效评价Synthesis and SAR of substituted tetrahydrocarbazole derivatives as new NPY-1 antagonists.

期刊:Bioorganic & medicinal chemistry letters发表年份:2006作者:Romano Di Fabio; Riccardo Giovannini; Barbara Bertani; Manuela Borriello; Andrea Bozzoli; Daniele Donati; Alessandro Falchi; Damiano Ghirlanda; Colin P Leslie; Angelo Pecunioso; Giovanna Rumboldt; Simone Spada

药效评价Nitrobenzylcarbamate prodrugs of cytotoxic acridines for potential use with nitroreductase gene-directed enzyme prodrug therapy.

期刊:Bioorganic & medicinal chemistry letters发表年份:2006作者:Christian Asche; Pascal Dumy; Danièle Carrez; Alain Croisy; Martine Demeunynck