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药效评价Identification of a novel spiropiperidine opioid receptor-like 1 antagonist class by a focused library approach featuring 3D-pharmacophore similarity.

期刊:Journal of medicinal chemistry发表年份:2006作者:Yasuhiro Goto; Sachie Arai-Otsuki; Yukari Tachibana; Daisuke Ichikawa; Satoshi Ozaki; Hiroyuki Takahashi; Yoshikazu Iwasawa; Osamu Okamoto; Shoki Okuda; Hisashi Ohta; Takeshi Sagara

药效评价Diarylacetylene piperidinyl amides as novel anxiolytics.

期刊:Bioorganic & medicinal chemistry letters发表年份:2006作者:Cheryl P Kordik; Chi Luo; Maryann Gutherman; Anil H Vaidya; Daniel I Rosenthal; Jeffrey J Crooke; Sandra L McKenney; Carlos R Plata-Salaman; Allen B Reitz

药效评价Discovery of 3-arylpropionic acids as potent agonists of sphingosine-1-phosphate receptor-1 (S1P1) with high selectivity against all other known S1P receptor subtypes.

期刊:Bioorganic & medicinal chemistry letters发表年份:2006作者:Lin Yan; Pei Huo; George Doherty; Lesile Toth; Jeffrey J Hale; Sander G Mills; Richard Hajdu; Carol A Keohane; Mark J Rosenbach; James A Milligan; Gan-Ju Shei; Gary Chrebet; James Bergstrom; Deborah Card; Elizabeth Quackenbush; Alexandra Wickham; Suz

药效评价Bioreactor systems for the production of biopharmaceuticals from animal cells.

期刊:Biotechnology and applied biochemistry发表年份:2006作者:James N Warnock; Mohamed Al-Rubeai