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药效评价Fentanyl-Type Antagonist of the μ-Opioid Receptor: Important Role of Axial Chirality in the Active Conformation.

期刊:Journal of medicinal chemistry发表年份:2024作者:Hironobu Arita; Ryoko Tanaka; Shuntaro Kikukawa; Tsukasa Tomizawa; Haruka Sakata; Masahiko Funada; Kenichi Tomiyama; Masaru Hashimoto; Tomohiko Tasaka; Hidetsugu Tabata; Kayo Nakamura; Kosho Makino; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahas

药效评价A novel, label-free, pre-equilibrium assay to determine the association and dissociation rate constants of therapeutic antibodies on living cells.

期刊:British journal of pharmacology发表年份:2024作者:Eric M Janezic; Alexander Doan; Elaine Mai; Daniel D Bravo; Jianyong Wang; Hok Seon Kim; Christoph Spiess; Kathryn Bewley; Adel ElSohly; Wei-Ching Liang; James T Koerber; Pascale Richalet; Marc Vanhove; Laetitia Comps-Agrar

药效评价Ubiquitin: Characterization of a Host Cell Protein Covalently Attached to a Monoclonal Antibody Product by LC-MS/MS.

期刊:Journal of pharmaceutical sciences发表年份:2024作者:Regina Kufer; Vincent Larraillet; Sabrina Thalhauser; Tobias Graf; Manuel Endesfelder; Stefanie Wohlrab

药效评价Platform development for high-throughput optimization of perfusion processes-Part II: Variation of perfusion rate strategies in microwell plates.

期刊:Biotechnology and bioengineering发表年份:2024作者:Marie Dorn; Ciara Lucas; Kerensa Klottrup-Rees; Ken Lee; Martina Micheletti