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药效评价Agonist-selective activation of individual G-proteins by muscarinic receptors.

期刊:Scientific reports发表年份:2024作者:Dominik Nelic; Nikolai Chetverikov; Martina Hochmalová; Christina Diaz; Vladimír Doležal; John Boulos; Jan Jakubík; Kirill Martemyanov; Alena Janoušková-Randáková

药效评价Intracellular Allosteric Antagonist of the Olfactory Receptor OR51E2.

期刊:Molecular pharmacology发表年份:2024作者:Tatjana Abaffy; Olivia Fu; Maira Harume-Nagai; Josh M Goldenberg; Victor Kenyon; Terry Kenakin

药效评价Identification of Acyl-Protein Thioesterase-1 as a Polysorbate-Degrading Host Cell Protein in a Monoclonal Antibody Formulation Using Activity-Based Protein Profiling.

期刊:Journal of pharmaceutical sciences发表年份:2024作者:Ernest Šprager; Jens Möller; Yuhsien Lin; Veronika Reisinger; Tomaž Bratkovič; Mojca Lunder; Jožica Vašl; Aleksander Krajnc

药效评价KCNE4-dependent modulation of Kv1.3 pharmacology.

期刊:Biochemical pharmacology发表年份:2024作者:Daniel Sastre; Magalí Colomer-Molera; Angela de Benito-Bueno; Carmen Valenzuela; Gregorio Fernández-Ballester; Antonio Felipe