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药效评价BRET- and fluorescence anisotropy-based assays for real-time monitoring of ligand binding to M2 muscarinic acetylcholine receptors.

期刊:Biochimica et biophysica acta. Molecular cell research发表年份:2021作者:Lukas Grätz; Tõnis Laasfeld; Anni Allikalt; Corinna G Gruber; Andrea Pegoli; Maris-Johanna Tahk; Mari-Liis Tsernant; Max Keller; Ago Rinken

药效评价Cell-based 3D bionic screening by mimicking the drug-receptor interaction environment in vivo.

期刊:Journal of materials chemistry. B发表年份:2021作者:Fen Wei; Xiaxi Zhang; Ping Cui; Xilan Gou; Sicen Wang

药效评价Tracking the Behavior of Monoclonal Antibody Product Quality Attributes Using a Multi-Attribute Method Workflow.

期刊:Journal of the American Society for Mass Spectrometry发表年份:2021作者:Craig Jakes; Silvia Millán-Martín; Sara Carillo; Kai Scheffler; Izabela Zaborowska; Jonathan Bones

药效评价Bicyclic Diazepinones as Dual Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels and the Norepinephrine Transporter.

期刊:Journal of medicinal chemistry发表年份:2021作者:José Luis Díaz; Félix Cuevas; Gonzalo Pazos; Paula Álvarez-Bercedo; Ana I Oliva; M Ángeles Sarmentero; Daniel Font; Agustín Jiménez-Aquino; María Morón; Adriana Port; Rosalía Pascual; Albert Dordal; Enrique Portillo-Salido; Raquel F Reinoso; José Mig