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药效评价Synthesis and evaluation of "Ama-Flash", a photocaged amatoxin prodrug for light-activated RNA Pol II inhibition and cell death.

期刊:Chemical communications (Cambridge, England)发表年份:2021作者:Kaveh Matinkhoo; Alla Pryyma; Antonio A W L Wong; David M Perrin

药效评价Rational Remodeling of Atypical Scaffolds for the Design of Photoswitchable Cannabinoid Receptor Tools.

期刊:Journal of medicinal chemistry发表年份:2021作者:Tao Hu; Guoxun Zheng; Dongxiang Xue; Simeng Zhao; Fei Li; Fang Zhou; Fei Zhao; Linshan Xie; Cuiping Tian; Tian Hua; Suwen Zhao; Yueming Xu; Guisheng Zhong; Zhi-Jie Liu; Alexandros Makriyannis; Raymond C Stevens; Houchao Tao

药效评价Detection of Isopeptide Bonds in Monoclonal Antibody Aggregates.

期刊:Pharmaceutical research发表年份:2021作者:Thomas Powell; Michael J Knight; Amanda Wood; John O'Hara; William Burkitt

药效评价Disentangling bias between Gq, GRK2, and arrestin3 recruitment to the M3 muscarinic acetylcholine receptor.

期刊:eLife发表年份:2021作者:Anja Flöser; Katharina Becker; Evi Kostenis; Gabriele König; Cornelius Krasel; Peter Kolb; Moritz Bünemann