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药效评价Macropinocytosis-Inducible Extracellular Vesicles Modified with Antimicrobial Protein CAP18-Derived Cell-Penetrating Peptides for Efficient Intracellular Delivery.

期刊:Molecular pharmaceutics发表年份:2021作者:Kosuke Noguchi; Momoko Obuki; Haruka Sumi; Merlin Klußmann; Kenta Morimoto; Shinya Nakai; Takuya Hashimoto; Daisuke Fujiwara; Ikuo Fujii; Eiji Yuba; Tomoka Takatani-Nakase; Ines Neundorf; Ikuhiko Nakase

药效评价Discovery of an M-Substituted N-Cyclopropylmethyl-7α-phenyl-6,14-endoethanotetrahydronorthebaine as a Selective, Potent, and Orally Active κ-Opioid Receptor Agonist with an Improved Central Nervous System Safety Profile.

期刊:Journal of medicinal chemistry发表年份:2021作者:Qian He; Yuanyuan Wei; Xiao Liu; Rongrong Ye; Linghui Kong; Zixiang Li; Shuang Jiang; Linqian Yu; Jingrui Chai; Qiong Xie; Wei Fu; Yujun Wang; Wei Li; Zhuibai Qiu; Jinggen Liu; Liming Shao

药效评价ST-2191, an Anellated Bismorpholino Derivative of Oxy-Fingolimod, Shows Selective S1P1 Agonist and Functional Antagonist Potency In Vitro and In Vivo.

期刊:Molecules (Basel, Switzerland)发表年份:2021作者:Bisera Stepanovska Tanturovska; Aleksandra Zivkovic; Faik Imeri; Thomas Homann; Burkhard Kleuser; Holger Stark; Andrea Huwiler

药效评价Post-Column Denaturation-Assisted Native Size-Exclusion Chromatography-Mass Spectrometry for Rapid and In-Depth Characterization of High Molecular Weight Variants in Therapeutic Monoclonal Antibodies.

期刊:Journal of the American Society for Mass Spectrometry发表年份:2021作者:Yuetian Yan; Tao Xing; Anita P Liu; Zhengqi Zhang; Shunhai Wang; Ning Li