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药效评价Genetic Up-Regulation or Pharmacological Activation of the Na+/Ca2+ Exchanger 1 (NCX1) Enhances Hippocampal-Dependent Contextual and Spatial Learning and Memory.

期刊:Molecular neurobiology发表年份:2020作者:Silvia Natale; Serenella Anzilotti; Tiziana Petrozziello; Roselia Ciccone; Angelo Serani; Lucrezia Calabrese; Beatrice Severino; Francesco Frecentese; Agnese Secondo; Anna Pannaccione; Ferdinando Fiorino; Ornella Cuomo; Antonio Vinciguerra; Lucia D'E

药效评价Small molecule somatostatin receptor subtype 4 (sst4) agonists are novel anti-inflammatory and analgesic drug candidates.

期刊:Neuropharmacology发表年份:2020作者:Éva Szőke; Mónika Bálint; Csaba Hetényi; Adrienn Markovics; Krisztián Elekes; Gábor Pozsgai; Tamás Szűts; György Kéri; László Őrfi; Zoltán Sándor; János Szolcsányi; Erika Pintér; Zsuzsanna Helyes

药效评价New insights on the arylpiperazinylalkyl pyridazinone ET1 as potent antinociceptive and anti-inflammatory agent.

期刊:European journal of pharmacology发表年份:2020作者:Francesco Μaione; Mariantonella Colucci; Federica Raucci; Giorgina Mangano; Francesca Marzoli; Nicola Mascolo; Letizia Crocetti; Maria Paola Giovannoni; Amalia Di Giannuario; Stefano Pieretti

药效评价Pharmacological characterisation of small molecule C5aR1 inhibitors in human cells reveals biased activities for signalling and function.

期刊:Biochemical pharmacology发表年份:2020作者:Xaria X Li; John D Lee; Nicholas L Massey; Carolyn Guan; Avril A B Robertson; Richard J Clark; Trent M Woodruff