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药效评价Venom alkaloids against Chagas disease parasite: search for effective therapies.

期刊:Scientific reports发表年份:2020作者:Rafael C M Costa Silva; Eduardo G P Fox; Fabio M Gomes; Daniel F Feijó; Isabela Ramos; Carolina M Koeller; Tatiana F R Costa; Nathalia S Rodrigues; Ana P Lima; Georgia C Atella; Kildare Miranda; Alejandra C Schoijet; Guillermo D Alonso; Ednildo de Al

药效评价Activation and Signaling Mechanism Revealed by Cannabinoid Receptor-Gi Complex Structures.

期刊:Cell发表年份:2020作者:Tian Hua; Xiaoting Li; Lijie Wu; Christos Iliopoulos-Tsoutsouvas; Yuxia Wang; Meng Wu; Ling Shen; Christina A Brust; Spyros P Nikas; Feng Song; Xiyong Song; Shuguang Yuan; Qianqian Sun; Yiran Wu; Shan Jiang; Travis W Grim; Othman Benchama; Edward L S

药效评价Affinity, potency, efficacy, selectivity, and molecular modeling of substituted fentanyls at opioid receptors.

期刊:Biochemical pharmacology发表年份:2020作者:Amy J Eshleman; Shanthi Nagarajan; Katherine M Wolfrum; John F Reed; Aaron Nilsen; Randy Torralva; Aaron Janowsky

药效评价In silico screening of GMQ-like compounds reveals guanabenz and sephin1 as new allosteric modulators of acid-sensing ion channel 3.

期刊:Biochemical pharmacology发表年份:2020作者:Gerard Callejo; Luke A Pattison; Jack C Greenhalgh; Sampurna Chakrabarti; Evangelia Andreopoulou; James R F Hockley; Ewan St John Smith; Taufiq Rahman