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药效评价Multi-target dopamine D3 receptor modulators: Actionable knowledge for drug design from molecular dynamics and machine learning.

期刊:European journal of medicinal chemistry发表年份:2020作者:Mariarosaria Ferraro; Sergio Decherchi; Alessio De Simone; Maurizio Recanatini; Andrea Cavalli; Giovanni Bottegoni

药效评价Tacrine-xanomeline and tacrine-iperoxo hybrid ligands: Synthesis and biological evaluation at acetylcholinesterase and M1 muscarinic acetylcholine receptors.

期刊:Bioorganic chemistry发表年份:2020作者:Marco Maspero; Daniela Volpato; Davide Cirillo; Natalia Yuan Chen; Regina Messerer; Christoph Sotriffer; Marco De Amici; Ulrike Holzgrabe; Clelia Dallanoce

药效评价Investigation of Inactive-State κ Opioid Receptor Homodimerization via Single-Molecule Microscopy Using New Antagonistic Fluorescent Probes.

期刊:Journal of medicinal chemistry发表年份:2020作者:Antonios Drakopoulos; Zsombor Koszegi; Yann Lanoiselée; Harald Hübner; Peter Gmeiner; Davide Calebiro; Michael Decker

药效评价Vestronidase alfa: Recombinant human β-glucuronidase as an enzyme replacement therapy for MPS VII.

期刊:Molecular genetics and metabolism发表年份:2020作者:Jaclyn Cadaoas; Gabrielle Boyle; Steven Jungles; Sean Cullen; Michel Vellard; Jeffrey H Grubb; Agnieszka Jurecka; William Sly; Emil Kakkis