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药效评价Annealing prion protein amyloid fibrils at high temperature results in extension of a proteinase K-resistant core.

期刊:The Journal of biological chemistry发表年份:2006作者:Olga V Bocharova; Natallia Makarava; Leonid Breydo; Maighdlin Anderson; Vadim V Salnikov; Ilia V Baskakov

药效评价Design, synthesis, and biological evaluation of the combinatorial library with a new spirodiketopiperazine scaffold. Discovery of novel potent and selective low-molecular-weight CCR5 antagonists.

期刊:Journal of medicinal chemistry发表年份:2006作者:Hiromu Habashita; Masaya Kokubo; Shin-ichi Hamano; Nobuyuki Hamanaka; Masaaki Toda; Shiro Shibayama; Hideaki Tada; Kenji Sagawa; Daikichi Fukushima; Kenji Maeda; Hiroaki Mitsuya

药效评价Immunohistochemical localization of a GHB receptor-like protein isolated from rat brain.

期刊:The Journal of comparative neurology发表年份:2006作者:Véronique Kemmel; Monique Miehe; Guy Roussel; Omar Taleb; Karine Nail-Boucherie; Christiane Marchand; Christine Stutz; Christian Andriamampandry; Dominique Aunis; Michel Maitre

药效评价Aripiprazole and its human metabolite are partial agonists at the human dopamine D2 receptor, but the rodent metabolite displays antagonist properties.

期刊:European journal of pharmacology发表年份:2006作者:Martyn D Wood; Claire Scott; Kirsten Clarke; Julie Westaway; Ceri H Davies; Charlie Reavill; Mark Hill; Claire Rourke; Michael Newson; Declan N C Jones; Ian T Forbes; Andrew Gribble