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代谢疾病Design, synthesis, and evaluation of novel 3-amino-4-hydrazine-cyclobut-3-ene-1,2-diones as potent and selective CXCR2 chemokine receptor antagonists.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Shilan Liu; Yinhui Liu; Hongmei Wang; Yili Ding; Hao Wu; Jingchao Dong; Angela Wong; Shu-Hui Chen; Ge Li; Manuel Chan; Nicole Sawyer; Francois G Gervais; Martin Henault; Stacia Kargman; Leanne L Bedard; Yongxin Han; Rick Friesen; Robert B Lobell; Dav

代谢疾病Peri-substituted hexahydro-indolones as novel, potent and selective human EP3 receptor antagonists.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Matthew O'Connell; Wayne Zeller; James Burgeson; Rama K Mishra; Jose Ramirez; Alex S Kiselyov; Thornorkell Andrésson; Mark E Gurney; Jasbir Singh

代谢疾病Islet neogenesis-associated protein pentadecapeptide (INGAP-PP): mechanisms involved in its effect upon beta-cell mass and function.

期刊:Regulatory peptides发表年份:2009作者:Viviana Madrid; Héctor Del Zotto; Bárbara Maiztegui; María A Raschia; María E Alzugaray; Antonio C Boschero; Helena C Barbosa; Luis E Flores; María I Borelli; Juan J Gagliardino

代谢疾病Cytotoxic, mutagenic and genotoxic effects of new anti-T. cruzi 5-phenylethenylbenzofuroxans. Contribution of phase I metabolites on the mutagenicity induction.

期刊:Toxicology letters发表年份:2009作者:Mauricio Cabrera; María Laura Lavaggi; Paola Hernández; Alicia Merlino; Alejandra Gerpe; Williams Porcal; Mariana Boiani; Ana Ferreira; Antonio Monge; Adela López de Cerain; Mercedes González; Hugo Cerecetto