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药效评价Bioactive Chemical Composition of Cannabis Extracts and Cannabinoid Receptors.

期刊:Molecules (Basel, Switzerland)发表年份:2020作者:Yi Yang; Rupali Vyawahare; Melissa Lewis-Bakker; Hance A Clarke; Albert H C Wong; Lakshmi P Kotra

药效评价Isoquinolinone derivatives as potent CNS multi-receptor D2/5-HT1A/5-HT2A/5-HT6/5-HT7 agents: Synthesis and pharmacological evaluation.

期刊:European journal of medicinal chemistry发表年份:2020作者:Jian Jin; Kunxiao Zhang; Fei Dou; Chao Hao; Yifang Zhang; Xudong Cao; Lanchang Gao; Jiaying Xiong; Xin Liu; Bi-Feng Liu; Guisen Zhang; Yin Chen

药效评价Discovery of Novel pERK1/2- or β-Arrestin-Preferring 5-HT1A Receptor-Biased Agonists: Diversified Therapeutic-like versus Side Effect Profile.

期刊:Journal of medicinal chemistry发表年份:2020作者:Joanna Sniecikowska; Monika Gluch-Lutwin; Adam Bucki; Anna Więckowska; Agata Siwek; Magdalena Jastrzebska-Wiesek; Anna Partyka; Daria Wilczyńska; Karolina Pytka; Gniewomir Latacz; Katarzyna Przejczowska-Pomierny; Elżbieta Wyska; Anna Wesołowska; Maci

药效评价Pharmacological characterisation of novel adenosine A3 receptor antagonists.

期刊:Scientific reports发表年份:2020作者:Kerry Barkan; Panagiotis Lagarias; Margarita Stampelou; Dimitrios Stamatis; Sam Hoare; Dewi Safitri; Karl-Norbert Klotz; Eleni Vrontaki; Antonios Kolocouris; Graham Ladds