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药效评价Striatal Kir2 K+ channel inhibition mediates the antidyskinetic effects of amantadine.

期刊:The Journal of clinical investigation发表年份:2020作者:Weixing Shen; Wenjie Ren; Shenyu Zhai; Ben Yang; Carlos G Vanoye; Ananya Mitra; Alfred L George; D James Surmeier

药效评价Discovery, Optimization, and Characterization of ML417: A Novel and Highly Selective D3 Dopamine Receptor Agonist.

期刊:Journal of medicinal chemistry发表年份:2020作者:Amy E Moritz; R Benjamin Free; Warren S Weiner; Emmanuel O Akano; Disha Gandhi; Ara Abramyan; Thomas M Keck; Marc Ferrer; Xin Hu; Noel Southall; Joseph Steiner; Jeffrey Aubé; Lei Shi; Kevin J Frankowski; David R Sibley

药效评价Discovery and structure-activity relationships study of positive allosteric modulators of the M3 muscarinic acetylcholine receptor.

期刊:Bioorganic & medicinal chemistry发表年份:2020作者:Hiroaki Tanaka; Kenji Negoro; Takanori Koike; Issei Tsukamoto; Kazuhiro Yokoyama; Jun Maeda; Yusuke Inagaki; Yukinori Shimoshige; Katsutoshi Ino; Kenichiro Ishizu; Taisuke Takahashi

药效评价Pharmacological Profile and Molecular Modeling of Cyclic Opioid Analogues Incorporating Various Phenylalanine Derivatives.

期刊:ChemMedChem发表年份:2020作者:Anna Adamska-Bartłomiejczyk; Piotr F J Lipiński; Justyna Piekielna-Ciesielska; Alicja Kluczyk; Anna Janecka