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代谢疾病Discovery of a novel azepine series of potent and selective 5-HT2C agonists as potential treatments for urinary incontinence.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Paul E Brennan; Gavin A Whitlock; Danny K H Ho; Kelly Conlon; Gordon McMurray

代谢疾病Discovery of a peroxisome proliferator activated receptor gamma (PPARgamma) modulator with balanced PPARalpha activity for the treatment of type 2 diabetes and dyslipidemia.

期刊:Journal of medicinal chemistry发表年份:2009作者:Weiguo Liu; Kun Liu; Harold B Wood; Margaret E McCann; Thomas W Doebber; Ching H Chang; Taro E Akiyama; Monica Einstein; Joel P Berger; Peter T Meinke

代谢疾病Metabolic labeling of sialic acids in living animals with alkynyl sugars.

期刊:Angewandte Chemie (International ed. in English)发表年份:2009作者:Pamela V Chang; Xing Chen; Chris Smyrniotis; Alexander Xenakis; Tianshun Hu; Carolyn R Bertozzi; Peng Wu

代谢疾病3-Acrylamide-4-aryloxyindoles: synthesis, biological evaluation and metabolic stability of potent and selective EP3 receptor antagonists.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Nian Zhou; Wayne Zeller; Jun Zhang; Emmanuel Onua; Alex S Kiselyov; Jose Ramirez; Gudrún Palsdottir; Gudrún Halldorsdottir; Thornorkell Andrésson; Mark E Gurney; Jasbir Singh