郑州微飒生物科技有限责任公司 咨询热线:0371-88821766
行业动态

行业动态

追踪行业前沿,洞察产业趋势

药效评价Computationally Guided Identification of Allosteric Agonists of the Metabotropic Glutamate 7 Receptor.

期刊:ACS chemical neuroscience发表年份:2019作者:Jose María Cid; Hilde Lavreysen; Gary Tresadern; Laura Pérez-Benito; Fulgencio Tovar; Alberto Fontana; Andrés A Trabanco

药效评价A comprehensive toxicological safety assessment of an extract of Ageratum conyzoides.

期刊:Regulatory toxicology and pharmacology : RTP发表年份:2019作者:Philip A Palmer; Jessica A Bryson; Amy E Clewell; John R Endres; Gábor Hirka; Adél Vértesi; Erzsébet Béres; Róbert Glávits; Ilona Pasics Szakonyiné

药效评价Development of a novel NURR1/NOT agonist from hit to lead and candidate for the potential treatment of Parkinson's disease.

期刊:Bioorganic & medicinal chemistry letters发表年份:2019作者:Dominique Lesuisse; André Malanda; Jean-François Peyronel; Yannick Evanno; Patrick Lardenois; Danielle De-Peretti; Pierre-Yves Abécassis; Pascal Barnéoud; Pascale Brunel; Marie-Claude Burgevin; Céline Cegarra; Florian Auger; Amélie Dommergue; Corinne

药效评价Comparative Docking to Distinct G Protein-Coupled Receptor Conformations Exclusively Yields Ligands with Agonist Efficacy.

期刊:Molecular pharmacology发表年份:2019作者:Magdalena M Scharf; Moritz Bünemann; Jillian G Baker; Peter Kolb