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药效评价Two New Neo-debromoaplysiatoxins-A Pair of Stereoisomers Exhibiting Potent Kv1.5 Ion Channel Inhibition Activities.

期刊:Marine drugs发表年份:2019作者:Ting-Ting Fan; Hui-Hui Zhang; Yang-Hua Tang; Fan-Zhong Zhang; Bing-Nan Han

药效评价N-Palmitoylglycine and other N-acylamides activate the lipid receptor G2A/GPR132.

期刊:Pharmacology research & perspectives发表年份:2019作者:James R Foster; Shohta Ueno; Mao Xiang Chen; Jenni Harvey; Simon J Dowell; Andrew J Irving; Andrew J Brown

药效评价Drug-receptor kinetics and sigma-1 receptor affinity differentiate clinically evaluated histamine H3 receptor antagonists.

期刊:Neuropharmacology发表年份:2019作者:Darren M Riddy; Anna E Cook; David M Shackleford; Tracie L Pierce; Elisabeth Mocaer; Clotilde Mannoury la Cour; Aurore Sors; William N Charman; Roger J Summers; Patrick M Sexton; Arthur Christopoulos; Christopher J Langmead

药效评价Label-free drug screening assay multiplexed with an orthogonal time-resolved fluorescence labeled assay.

期刊:Analytical biochemistry发表年份:2019作者:László Kiss; Attila Cselenyák; András Visegrády