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药效评价Targeting the CaVα-CaVβ interaction yields an antagonist of the N-type CaV2.2 channel with broad antinociceptive efficacy.

期刊:Pain发表年份:2019作者:Rajesh Khanna; Jie Yu; Xiaofang Yang; Aubin Moutal; Aude Chefdeville; Vijay Gokhale; Zunaira Shuja; Lindsey A Chew; Shreya S Bellampalli; Shizhen Luo; Liberty François-Moutal; Maria J Serafini; Taehwan Ha; Samantha Perez-Miller; Ki Duk Park; Amol M P

药效评价7-Amino-2-aryl/hetero-aryl-5-oxo-5,8-dihydro[1,2,4]triazolo[1,5-a]pyridine-6-carbonitriles: Synthesis and adenosine receptor binding studies.

期刊:Chemical biology & drug design发表年份:2019作者:Khasim Shaik; Pran Kishore Deb; Raghu Prasad Mailavaram; Balakumar Chandrasekaran; Sonja Kachler; Karl-Norbert Klotz; Abdul Muttaleb Yousef Jaber

药效评价Histidine at position 462 determines the low quinine sensitivity of ether-à-go-go channel superfamily member Kv 12.1.

期刊:British journal of pharmacology发表年份:2019作者:Marlen Dierich; Willem B van Ham; Anna Stary-Weinzinger; Michael G Leitner

药效评价Efficient Site-Specific Antibody-Drug Conjugation by Engineering a Nature-Derived Recognition Tag for Microbial Transglutaminase.

期刊:Chembiochem : a European journal of chemical biology发表年份:2019作者:Aileen Ebenig; Norbert Egon Juettner; Lukas Deweid; Olga Avrutina; Hans-Lothar Fuchsbauer; Harald Kolmar