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药效评价Design and synthesis of cyclopropane-based conformationally restricted GABA analogues as selective inhibitors for betaine/GABA transporter 1.

期刊:Bioorganic & medicinal chemistry letters发表年份:2018作者:Akihiro Suemasa; Mizuki Watanabe; Takaaki Kobayashi; Hiroe Suzuki; Hayato Fukuda; Masabumi Minami; Satoshi Shuto

药效评价Pharmacological Characterization of Dezocine, a Potent Analgesic Acting as a κ Partial Agonist and μ Partial Agonist.

期刊:Scientific reports发表年份:2018作者:Yu-Hua Wang; Jing-Rui Chai; Xue-Jun Xu; Ru-Feng Ye; Gui-Ying Zan; George Yun-Kun Liu; Jian-Dong Long; Yan Ma; Xiang Huang; Zhi-Chao Xiao; Hu Dong; Yu-Jun Wang

药效评价Recombinant human follicle stimulating hormone purification by a short peptide affinity chromatography.

期刊:Journal of peptide science : an official publication of the European Peptide Society发表年份:2018作者:Juan M Gurevich Messina; Silvana L Giudicessi; María C Martínez Ceron; Nicolás Urtasun; Guillermina Forno; Laura Mauro; Osvaldo Cascone; Silvia A Camperi

药效评价Preassembled GPCR signaling complexes mediate distinct cellular responses to ultralow ligand concentrations.

期刊:Science signaling发表年份:2018作者:Srgjan Civciristov; Andrew M Ellisdon; Ryan Suderman; Cindy K Pon; Bronwyn A Evans; Oded Kleifeld; Steven J Charlton; William S Hlavacek; Meritxell Canals; Michelle L Halls