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药效评价PF-06526290 can both enhance and inhibit conduction through voltage-gated sodium channels.

期刊:British journal of pharmacology发表年份:2018作者:Lingxin Wang; Shannon G Zellmer; David M Printzenhoff; Neil A Castle

药效评价A New Fluorogenic Small-Molecule Labeling Tool for Surface Diffusion Analysis and Advanced Fluorescence Imaging of β-Site Amyloid Precursor Protein-Cleaving Enzyme 1 Based on Silicone Rhodamine: SiR-BACE1.

期刊:Journal of medicinal chemistry发表年份:2018作者:Sandra Karch; Johannes Broichhagen; Julia Schneider; Daniel Böning; Stephanie Hartmann; Benjamin Schmid; Philipp Tripal; Ralf Palmisano; Christian Alzheimer; Kai Johnsson; Tobias Huth

药效评价Genistein Enhances or Reduces Glycosaminoglycan Quantity in a Cell Type-Specific Manner.

期刊:Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology发表年份:2018作者:Ying Lan; Xiulian Li; Xuebo Liu; Cui Hao; Ni Song; Sumei Ren; Wei Wang; Ningchuan Feng; Lijuan Zhang

药效评价Methylation Products of 6β- N-Heterocyclic Substituted Naltrexamine Derivatives as Potential Peripheral Opioid Receptor Modulators.

期刊:ACS chemical neuroscience发表年份:2018作者:Yi Zheng; Samuel Obeng; Huiqun Wang; David L Stevens; Essie Komla; Dana E Selley; William L Dewey; Hamid I Akbarali; Yan Zhang