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药效评价Docking Screens for Dual Inhibitors of Disparate Drug Targets for Parkinson's Disease.

期刊:Journal of medicinal chemistry发表年份:2018作者:Mariama Jaiteh; Alexey Zeifman; Marcus Saarinen; Per Svenningsson; Jose Bréa; Maria Isabel Loza; Jens Carlsson

药效评价Characterization of methanthelinium binding and function at human M1-M5 muscarinic acetylcholine receptors.

期刊:Naunyn-Schmiedeberg's archives of pharmacology发表年份:2018作者:Matthias Irmen; Janine Holze; Theresa Bödefeld; Christian Tränkle

药效评价Neonatal Fc receptor antagonist efgartigimod safely and sustainably reduces IgGs in humans.

期刊:The Journal of clinical investigation发表年份:2018作者:Peter Ulrichts; Antonio Guglietta; Torsten Dreier; Tonke van Bragt; Valérie Hanssens; Erik Hofman; Bernhardt Vankerckhoven; Peter Verheesen; Nicolas Ongenae; Valentina Lykhopiy; F Javier Enriquez; JunHaeng Cho; Raimund J Ober; E Sally Ward; Hans de H

药效评价Discovery of artificial VIPR2-antagonist peptides possessing receptor- and ligand-selectivity.

期刊:Biochemical and biophysical research communications发表年份:2018作者:Kotaro Sakamoto; Ryokichi Koyama; Yusuke Kamada; Masanori Miwa; Akiyoshi Tani