药效评价2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist.
期刊:Journal of medicinal chemistry发表年份:2006作者:Cécile Enguehard-Gueiffier; Harald Hübner; Ahmed El Hakmaoui; Hassan Allouchi; Peter Gmeiner; Antonio Argiolas; Maria Rosaria Melis; Alain Gueiffier