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代谢疾病Oxadiazole-diarylpyrazole 4-carboxamides as cannabinoid CB1 receptor ligands.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Suk Ho Lee; Hee Jeong Seo; Min Ju Kim; Suk Youn Kang; Kwang-Seop Song; Sung-Han Lee; Myung Eun Jung; Jeongmin Kim; Jinhwa Lee

代谢疾病(1R, 3S)-(-)-trans-PAT: a novel full-efficacy serotonin 5-HT2C receptor agonist with 5-HT2A and 5-HT2B receptor inverse agonist/antagonist activity.

期刊:European journal of pharmacology发表年份:2009作者:Raymond G Booth; Lijuan Fang; Yingsu Huang; Andrzej Wilczynski; Sashikala Sivendran

代谢疾病Improving metabolic stability by glycosylation: bifunctional peptide derivatives that are opioid receptor agonists and neurokinin 1 receptor antagonists.

期刊:Journal of medicinal chemistry发表年份:2009作者:Takashi Yamamoto; Padma Nair; Neil E Jacobsen; Josef Vagner; Vinod Kulkarni; Peg Davis; Shou-Wu Ma; Edita Navratilova; Henry I Yamamura; Todd W Vanderah; Frank Porreca; Josephine Lai; Victor J Hruby

代谢疾病Glucagon-like peptide 1/glucagon receptor dual agonism reverses obesity in mice.

期刊:Diabetes发表年份:2009作者:Alessandro Pocai; Paul E Carrington; Jennifer R Adams; Michael Wright; George Eiermann; Lan Zhu; Xiaobing Du; Aleksandr Petrov; Michael E Lassman; Guoqiang Jiang; Franklin Liu; Corey Miller; Laurie M Tota; Gaochao Zhou; Xiaoping Zhang; Michael M Soun