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药效评价Placement of Hydroxy Moiety on Pendant of Peptidomimetic Scaffold Modulates Mu and Kappa Opioid Receptor Efficacy.

期刊:ACS chemical neuroscience发表年份:2017作者:Aubrie A Harland; Irina D Pogozheva; Nicholas W Griggs; Tyler J Trask; John R Traynor; Henry I Mosberg

药效评价Molecular Switches of Allosteric Modulation of the Metabotropic Glutamate 2 Receptor.

期刊:Structure (London, England : 1993)发表年份:2017作者:Laura Pérez-Benito; Maarten L J Doornbos; Arnau Cordomí; Luc Peeters; Hilde Lavreysen; Leonardo Pardo; Gary Tresadern

药效评价Isoform-Specific Biased Agonism of Histamine H3 Receptor Agonists.

期刊:Molecular pharmacology发表年份:2017作者:Darren M Riddy; Anna E Cook; Natalie A Diepenhorst; Sanja Bosnyak; Ryan Brady; Clotilde Mannoury la Cour; Elisabeth Mocaer; Roger J Summers; William N Charman; Patrick M Sexton; Arthur Christopoulos; Christopher J Langmead

药效评价Effector-attenuating Substitutions That Maintain Antibody Stability and Reduce Toxicity in Mice.

期刊:The Journal of biological chemistry发表年份:2017作者:Megan Lo; Hok Seon Kim; Raymond K Tong; Travis W Bainbridge; Jean-Michel Vernes; Yin Zhang; Yuwen Linda Lin; Shan Chung; Mark S Dennis; Y Joy Yu Zuchero; Ryan J Watts; Jessica A Couch; Y Gloria Meng; Jasvinder K Atwal; Randall J Brezski; Christoph Sp