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药效评价Pharmaco-toxicological effects of the novel third-generation fluorinate synthetic cannabinoids, 5F-ADBINACA, AB-FUBINACA, and STS-135 in mice. In vitro and in vivo studies.

期刊:Human psychopharmacology发表年份:2017作者:Isabella Canazza; Andrea Ossato; Fabrizio Vincenzi; Adolfo Gregori; Fabiana Di Rosa; Federica Nigro; Alessandro Rimessi; Paolo Pinton; Katia Varani; Pier Andrea Borea; Matteo Marti

药效评价A Novel Selective Inverse Agonist of the CB2 Receptor as a Radiolabeled Tool Compound for Kinetic Binding Studies.

期刊:Molecular pharmacology发表年份:2017作者:Andrea Martella; Huub Sijben; Arne C Rufer; Uwe Grether; Juergen Fingerle; Christoph Ullmer; Thomas Hartung; Adriaan P IJzerman; Mario van der Stelt; Laura H Heitman

药效评价A common mechanism for CFTR potentiators.

期刊:The Journal of general physiology发表年份:2017作者:Han-I Yeh; Yoshiro Sohma; Katja Conrath; Tzyh-Chang Hwang

药效评价Novel 5-HT7R antagonists, arylsulfonamide derivatives of (aryloxy)propyl piperidines: Add-on effect to the antidepressant activity of SSRI and DRI, and pro-cognitive profile.

期刊:Bioorganic & medicinal chemistry发表年份:2017作者:Vittorio Canale; Anna Partyka; Rafał Kurczab; Martyna Krawczyk; Tomasz Kos; Grzegorz Satała; Bartłomiej Kubica; Magdalena Jastrzębska-Więsek; Anna Wesołowska; Andrzej J Bojarski; Piotr Popik; Paweł Zajdel