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药效评价A novel TRPM8 agonist relieves dry eye discomfort.

期刊:BMC ophthalmology发表年份:2017作者:Jee Myung Yang; Fengxian Li; Qin Liu; Marco Rüedi; Edward Tak Wei; Michael Lentsman; Hyo Seok Lee; Won Choi; Seong Jin Kim; Kyung Chul Yoon

药效评价Inhibition of the potassium channel KCa3.1 by senicapoc reverses tactile allodynia in rats with peripheral nerve injury.

期刊:European journal of pharmacology发表年份:2017作者:Roland G W Staal; Tanzilya Khayrullina; Hong Zhang; Scott Davis; Shaun M Fallon; Manuel Cajina; Megan E Nattini; Andrew Hu; Hua Zhou; Suresh Babu Poda; Stevin Zorn; Gamini Chandrasena; Elena Dale; Brian Cambpell; Lars Christian Biilmann Rønn; Gordon

药效评价Heat-shock protein 90 (Hsp90) promotes opioid-induced anti-nociception by an ERK mitogen-activated protein kinase (MAPK) mechanism in mouse brain.

期刊:The Journal of biological chemistry发表年份:2017作者:Wei Lei; Nathan Mullen; Sarah McCarthy; Courtney Brann; Philomena Richard; James Cormier; Katie Edwards; Edward J Bilsky; John M Streicher

药效评价KK-92A, a novel GABAB receptor positive allosteric modulator, attenuates nicotine self-administration and cue-induced nicotine seeking in rats.

期刊:Psychopharmacology发表年份:2017作者:Xia Li; Emmanuel Sturchler; Katarzyna Kaczanowska; Michael Cameron; M G Finn; Patrick Griffin; Patricia McDonald; Athina Markou