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药效评价Extrapyramidal side effects of antipsychotics are linked to their association kinetics at dopamine D2 receptors.

期刊:Nature communications发表年份:2017作者:David A Sykes; Holly Moore; Lisa Stott; Nicholas Holliday; Jonathan A Javitch; J Robert Lane; Steven J Charlton

药效评价Synthesis, Pharmacology, and Molecular Docking Studies on 6-Desoxo-N-methylmorphinans as Potent μ-Opioid Receptor Agonists.

期刊:Journal of medicinal chemistry发表年份:2017作者:Maria Dumitrascuta; Tanila Ben Haddou; Elena Guerrieri; Stefan M Noha; Lea Schläfer; Helmut Schmidhammer; Mariana Spetea

药效评价An Aliphatic Ester Diisopropyl Sebacate Exhibited an Adjuvant Effect on Fluorescein Isothiocyanate-Induced Contact Hypersensitivity Mouse Models.

期刊:Biological & pharmaceutical bulletin发表年份:2018作者:Kohta Kurohane; Ayako Kimura; Rie Terasawa; Kamiyu Kobayashi; Wakana Suzuki; Takeshi Matsuoka; Yasuyuki Imai

药效评价A Complementary Scale of Biased Agonism for Agonists with Differing Maximal Responses.

期刊:Scientific reports发表年份:2017作者:Javier Burgueño; Marta Pujol; Xavier Monroy; David Roche; Maria Jose Varela; Manuel Merlos; Jesús Giraldo