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药效评价Design and Synthesis of Benzimidazoles As Novel Corticotropin-Releasing Factor 1 Receptor Antagonists.

期刊:Journal of medicinal chemistry发表年份:2016作者:Michiyo Mochizuki; Masakuni Kori; Katsumi Kobayashi; Takahiko Yano; Yuu Sako; Maiko Tanaka; Naoyuki Kanzaki; Albert C Gyorkos; Christopher P Corrette; Suk Young Cho; Scott A Pratt; Kazuyoshi Aso

药效评价Equilibrium and kinetic selectivity profiling on the human adenosine receptors.

期刊:Biochemical pharmacology发表年份:2016作者:Dong Guo; Gabrielle S Dijksteel; Tirsa van Duijl; Maxime Heezen; Laura H Heitman; Adriaan P IJzerman

药效评价Both Reversible Self-Association and Structural Changes Underpin Molecular Viscoelasticity of mAb Solutions.

期刊:Journal of pharmaceutical sciences发表年份:2016作者:Prasad S Sarangapani; Justin Weaver; Arun Parupudi; Tabot M D Besong; Gary G Adams; Stephen E Harding; Prakash Manikwar; Maria M Castellanos; Steven M Bishop; Jai A Pathak

药效评价Role of the Second Extracellular Loop of the Adenosine A1 Receptor on Allosteric Modulator Binding, Signaling, and Cooperativity.

期刊:Molecular pharmacology发表年份:2016作者:Anh T N Nguyen; Elizabeth A Vecchio; Trayder Thomas; Toan D Nguyen; Luigi Aurelio; Peter J Scammells; Paul J White; Patrick M Sexton; Karen J Gregory; Lauren T May; Arthur Christopoulos