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药效评价Controlled superficial assembly of DNA-amorphous calcium phosphate nanocomposite spheres for surface-mediated gene delivery.

期刊:Colloids and surfaces. B, Biointerfaces发表年份:2016作者:Ayako Oyane; Hiroko Araki; Maki Nakamura; Yoshiki Shimizu; Quazi T H Shubhra; Atsuo Ito; Hideo Tsurushima

药效评价Identification of a small-molecule ligand that activates the neuropeptide receptor GPR171 and increases food intake.

期刊:Science signaling发表年份:2016作者:Jonathan H Wardman; Ivone Gomes; Erin N Bobeck; Jennifer A Stockert; Abhijeet Kapoor; Paola Bisignano; Achla Gupta; Mihaly Mezei; Sanjai Kumar; Marta Filizola; Lakshmi A Devi

药效评价Characterization of methadone as a β-arrestin-biased μ-opioid receptor agonist.

期刊:Molecular pain发表年份:2016作者:Seira Doi; Tomohisa Mori; Naoki Uzawa; Takamichi Arima; Tomoyuki Takahashi; Masashi Uchida; Ayaka Yawata; Michiko Narita; Yasuhito Uezono; Tsutomu Suzuki; Minoru Narita

药效评价4-Phenylpyridin-2-one Derivatives: A Novel Class of Positive Allosteric Modulator of the M1 Muscarinic Acetylcholine Receptor.

期刊:Journal of medicinal chemistry发表年份:2016作者:Shailesh N Mistry; Manuela Jörg; Herman Lim; Natalie B Vinh; Patrick M Sexton; Ben Capuano; Arthur Christopoulos; J Robert Lane; Peter J Scammells