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药效评价4-amino-6-alkyloxy-2-alkylthiopyrimidine derivatives as novel non-nucleoside agonists for the adenosine A1 receptor.

期刊:Chemical biology & drug design发表年份:2016作者:Barbara Cosimelli; Giovanni Greco; Sonia Laneri; Ettore Novellino; Antonia Sacchi; Maria Letizia Trincavelli; Chiara Giacomelli; Sabrina Taliani; Federico Da Settimo; Claudia Martini

药效评价Scintillation proximity assay (SPA) as a new approach to determine a ligand's kinetic profile. A case in point for the adenosine A1 receptor.

期刊:Purinergic signalling发表年份:2016作者:Lizi Xia; Henk de Vries; Ad P IJzerman; Laura H Heitman

药效评价Ligand Binding Ensembles Determine Graded Agonist Efficacies at a G Protein-coupled Receptor.

期刊:The Journal of biological chemistry发表年份:2016作者:Andreas Bock; Marcel Bermudez; Fabian Krebs; Carlo Matera; Brian Chirinda; Dominique Sydow; Clelia Dallanoce; Ulrike Holzgrabe; Marco De Amici; Martin J Lohse; Gerhard Wolber; Klaus Mohr

药效评价Ultrastructural and morphological changes in Leishmania (Viannia) braziliensis treated with synthetic chalcones.

期刊:Experimental parasitology发表年份:2016作者:Tatiane F P de Mello; Bruna M Cardoso; Heriberto R Bitencourt; Lucélia Donatti; Sandra M A Aristides; Maria V C Lonardoni; Thais G V Silveira