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药效评价Novel Irreversible Agonists Acting at the A1 Adenosine Receptor.

期刊:Journal of medicinal chemistry发表年份:2016作者:Manuela Jörg; Alisa Glukhova; Alaa Abdul-Ridha; Elizabeth A Vecchio; Anh T N Nguyen; Patrick M Sexton; Paul J White; Lauren T May; Arthur Christopoulos; Peter J Scammells

药效评价A novel substituted aminoquinoline selectively targets voltage-sensitive sodium channel isoforms and NMDA receptor subtypes and alleviates chronic inflammatory and neuropathic pain.

期刊:European journal of pharmacology发表年份:2016作者:Boris Tabakoff; Wenhua Ren; Lauren Vanderlinden; Lawrence D Snell; Christopher J Matheson; Ze-Jun Wang; Rock Levinson; C Thetford Smothers; John J Woodward; Yumiko Honse; David Lovinger; Anthony M Rush; William A Sather; Daniel L Gustafson; Paula L H

药效评价Total synthesis and structure-activity relationship studies of a series of selective G protein inhibitors.

期刊:Nature chemistry发表年份:2016作者:Xiao-Feng Xiong; Hang Zhang; Christina R Underwood; Kasper Harpsøe; Thomas J Gardella; Mie F Wöldike; Michael Mannstadt; David E Gloriam; Hans Bräuner-Osborne; Kristian Strømgaard

药效评价In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations.

期刊:European journal of pharmacology发表年份:2016作者:Federica Ferrari; Maria Camilla Cerlesi; Davide Malfacini; Laila Asth; Elaine C Gavioli; Blair V Journigan; Uma Gayathri Kamakolanu; Michael E Meyer; Dennis Yasuda; Willma E Polgar; Anna Rizzi; Remo Guerrini; Chiara Ruzza; Nurulain T Zaveri; Girolamo