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药效评价Novel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity.

期刊:Journal of medicinal chemistry发表年份:2016作者:Mu-Fa Zou; Thomas M Keck; Vivek Kumar; Prashant Donthamsetti; Mayako Michino; Caitlin Burzynski; Catherine Schweppe; Alessandro Bonifazi; R Benjamin Free; David R Sibley; Aaron Janowsky; Lei Shi; Jonathan A Javitch; Amy Hauck Newman

药效评价Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT6 Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with Alzheimer's Disease.

期刊:ACS chemical neuroscience发表年份:2016作者:Katarzyna Grychowska; Grzegorz Satała; Tomasz Kos; Anna Partyka; Evelina Colacino; Severine Chaumont-Dubel; Xavier Bantreil; Anna Wesołowska; Maciej Pawłowski; Jean Martinez; Philippe Marin; Gilles Subra; Andrzej J Bojarski; Frédéric Lamaty; Piotr Po

药效评价Ligand Specific Efficiency (LSE) Index for PET Tracer Optimization.

期刊:ChemMedChem发表年份:2016作者:Yves P Auberson; Emmanuelle Briard; David Sykes; John Reilly; Mark Healy

药效评价6β-N-Heterocyclic Substituted Naltrexamine Derivative BNAP: A Peripherally Selective Mixed MOR/KOR Ligand.

期刊:ACS chemical neuroscience发表年份:2016作者:Dwight A Williams; Yi Zheng; Bethany G David; Yunyun Yuan; Saheem A Zaidi; David L Stevens; Krista L Scoggins; Dana E Selley; William L Dewey; Hamid I Akbarali; Yan Zhang