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药效评价The role of kinetic context in apparent biased agonism at GPCRs.

期刊:Nature communications发表年份:2016作者:Carmen Klein Herenbrink; David A Sykes; Prashant Donthamsetti; Meritxell Canals; Thomas Coudrat; Jeremy Shonberg; Peter J Scammells; Ben Capuano; Patrick M Sexton; Steven J Charlton; Jonathan A Javitch; Arthur Christopoulos; J Robert Lane

药效评价Optimization of a Novel Quinazolinone-Based Series of Transient Receptor Potential A1 (TRPA1) Antagonists Demonstrating Potent in Vivo Activity.

期刊:Journal of medicinal chemistry发表年份:2016作者:Laurie B Schenkel; Philip R Olivieri; Alessandro A Boezio; Holly L Deak; Renee Emkey; Russell F Graceffa; Hakan Gunaydin; Angel Guzman-Perez; Josie H Lee; Yohannes Teffera; Weiya Wang; Beth D Youngblood; Violeta L Yu; Maosheng Zhang; Narender R Gavva

药效评价Risk assessment of a cold argon plasma jet in respect to its mutagenicity.

期刊:Mutation research. Genetic toxicology and environmental mutagenesis发表年份:2016作者:K Wende; S Bekeschus; A Schmidt; L Jatsch; S Hasse; K D Weltmann; K Masur; T von Woedtke

药效评价Structure-guided development of dual β2 adrenergic/dopamine D2 receptor agonists.

期刊:Bioorganic & medicinal chemistry发表年份:2016作者:Dietmar Weichert; Markus Stanek; Harald Hübner; Peter Gmeiner