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药效评价The A- and B-type muscarinic acetylcholine receptors from Drosophila melanogaster couple to different second messenger pathways.

期刊:Biochemical and biophysical research communications发表年份:2015作者:Guilin R Ren; Jonas Folke; Frank Hauser; Shizhong Li; Cornelis J P Grimmelikhuijzen

药效评价Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists.

期刊:Molecular pharmacology发表年份:2015作者:Darren M Riddy; Celine Valant; Patricia Rueda; William N Charman; Patrick M Sexton; Roger J Summers; Arthur Christopoulos; Christopher J Langmead

药效评价Resin-acid derivatives as potent electrostatic openers of voltage-gated K channels and suppressors of neuronal excitability.

期刊:Scientific reports发表年份:2015作者:Nina E Ottosson; Xiongyu Wu; Andreas Nolting; Urban Karlsson; Per-Eric Lund; Katinka Ruda; Stefan Svensson; Peter Konradsson; Fredrik Elinder

药效评价Selective Allosteric Antagonists for the G Protein-Coupled Receptor GPRC6A Based on the 2-Phenylindole Privileged Structure Scaffold.

期刊:Journal of medicinal chemistry发表年份:2015作者:Henrik Johansson; Michael Worch Boesgaard; Lenea Nørskov-Lauritsen; Inna Larsen; Sebastiaan Kuhne; David E Gloriam; Hans Bräuner-Osborne; Daniel Sejer Pedersen