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药效评价CB2 cannabinoid receptor agonist enantiomers HU-433 and HU-308: An inverse relationship between binding affinity and biological potency.

期刊:Proceedings of the National Academy of Sciences of the United States of America发表年份:2015作者:Reem Smoum; Saja Baraghithy; Mukesh Chourasia; Aviva Breuer; Naama Mussai; Malka Attar-Namdar; Natalya M Kogan; Bitya Raphael; Daniele Bolognini; Maria G Cascio; Pietro Marini; Roger G Pertwee; Avital Shurki; Raphael Mechoulam; Itai Bab

药效评价Efficient entry of cell-penetrating peptide nona-arginine into adherent cells involves a transient increase in intracellular calcium.

期刊:The Biochemical journal发表年份:2015作者:Kamran Melikov; Ann Hara; Kwabena Yamoah; Elena Zaitseva; Eugene Zaitsev; Leonid V Chernomordik

药效评价Structure-Activity Relationships of the Peptide Kappa Opioid Receptor Antagonist Zyklophin.

期刊:Journal of medicinal chemistry发表年份:2015作者:Anand A Joshi; Thomas F Murray; Jane V Aldrich

药效评价Pharmacological Analysis and Structure Determination of 7-Methylcyanopindolol-Bound β1-Adrenergic Receptor.

期刊:Molecular pharmacology发表年份:2015作者:Tomomi Sato; Jillian Baker; Tony Warne; Giles A Brown; Andrew G W Leslie; Miles Congreve; Christopher G Tate